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| RVMDRVMDRevolution Medicines, Inc. | Revolution Medicines, Inc. | $186.99 | $40.1B |
| TNGXTNGXTango Therapeutics, Inc. | Tango Therapeutics, Inc. | $23.34 | $3.9B |
| IDYAIDYAIDEAYA Biosciences, Inc. | IDEAYA Biosciences, Inc. | $34.71 | $3.3B |
| NUVBNUVBNuvation Bio Inc. | Nuvation Bio Inc. | $4.57 | $1.6B |
| ORICORICORIC Pharmaceuticals, Inc. | ORIC Pharmaceuticals, Inc. | $13.17 | $1.4B |
| AVBPAVBPArriVent BioPharma, Inc. | ArriVent BioPharma, Inc. | $21.00 | $1.0B |
| VSTMVSTMVerastem, Inc. | Verastem, Inc. | $10.04 | $909.3M |
| KURAKURAKura Oncology, Inc. | Kura Oncology, Inc. | $9.61 | $854.9M |
| CRISCRISCuris, Inc. | Curis, Inc. | $0.39 | $753.3K |